Mitkin, Oleg D. : rechercher sur Z-Library

Le plus grand référentiel d'articles scientifiques au monde. 70,000,000+ d'articles gratuitement.

Don't use scam websites

Livres
Articles (38)
Les plus populaires
Liste
- Liste
- Tableau

1

Synthesis and Biological Evaluation of Novel 5,8-Disubstituted-2-methyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b] indoles as 5-HT6 and H1 Receptors Antagonists

Alexandre V. Ivachtchenko, Eugene B. Frolov, Oleg D. Mitkin, Volodymyr M. Kysil, Alexander V. Khvat, Sergey E. Tkachenko

Journal:

Archiv der Pharmazie

Année:

2009

Langue:

english

Fichier:

PDF, 426 KB

english, 2009

2

ChemInform Abstract: Indoles from 3-Nitropyridinium Salts. Part 12. An Extension of the Transformation Method on 5-Substituted Indoles.

Oleg D. Mitkin, Roman V. Kombarov, Marina A. Yurovskaya

Journal:

Année:

2001

Fichier:

PDF, 31 KB

2001

3

ChemInform Abstract: 8-Sulfonyl-Substituted Tetrahydro-1H-pyrido[4,3-b]indoles as 5-HT6 Receptor Antagonists.

Alexandre V. Ivachtchenko, Oleg D. Mitkin, Sergey E. Tkachenko, Ilya M. Okun, Volodymyr M. Kysil

Journal:

Année:

2010

Fichier:

PDF, 19 KB

2010

4

ChemInform Abstract: Bromination of Indomethacin.

Alexandre V. Ivachtchenko, Pavel M. Yamanushkin, Oleg D. Mitkin, Oleg I. Kiselev

Journal:

Année:

2010

Fichier:

PDF, 22 KB

2010

5

ChemInform Abstract: 2-Substituted 5,6-Dimethyl-3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidines: New Series of Highly Potent and Specific Serotonin 5-HT6 Receptor Antagonists.

Alexandre V. Ivachtchenko, Elena S. Golovina, Madina G. Kadieva, Angela G. Koryakova, Oleg D. Mitkin, Sergey E. Tkachenko, Volodymyr M. Kysil, Ilya Okun

Journal:

Année:

2011

Fichier:

PDF, 22 KB

2011

6

Bromination of indomethacin

Alexandre V. Ivachtchenko, Pavel M. Yamanushkin, Oleg D. Mitkin, Oleg I. Kiselev

Journal:

Mendeleev Communications

Année:

2010

Langue:

english

Fichier:

PDF, 217 KB

english, 2010

7

Synthesis and biological study of 3-(phenylsulfonyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidines as potent and selective serotonin 5-HT6 receptor antagonists

Alexandre V. Ivachtchenko, Elena S. Golovina, Madina G. Kadieva, Angela G. Koryakova, Sergiy M. Kovalenko, Oleg D. Mitkin, Ilya M. Okun, Irina M. Ravnyeyko, Sergey E. Tkachenko, Oleg V. Zaremba

Journal:

Bioorganic & Medicinal Chemistry

Année:

2010

Langue:

english

Fichier:

PDF, 511 KB

english, 2010

8

Synthesis and biological evaluation of novel γ-carboline analogues of Dimebon as potent 5-HT6 receptor antagonists

Alexandre V. Ivachtchenko, Eugene B. Frolov, Oleg D. Mitkin, Volodymyr M. Kysil, Alexander V. Khvat, Ilya M. Okun, Sergey E. Tkachenko

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2009

Langue:

english

Fichier:

PDF, 457 KB

english, 2009

9

Synthesis and biological activity of 5-styryl and 5-phenethyl-substituted 2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indoles

Alexandre V. Ivachtchenko, Eugen B. Frolov, Oleg D. Mitkin, Sergei E. Tkachenko, Ilya M. Okun, Alex V. Khvat

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2010

Langue:

english

Fichier:

PDF, 379 KB

english, 2010

10

Synthesis of cycloalkane-annelated 3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidines and their evaluation as 5-HT6 receptor antagonists

Alexandre V. Ivachtchenko, Dmitri E. Dmitriev, Elena S. Golovina, Elena S. Dubrovskaya, Madina G. Kadieva, Angela G. Koryakova, Volodymyr M. Kysil, Oleg D. Mitkin, Sergey E. Tkachenko, Ilya M. Okun, A

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2010

Langue:

english

Fichier:

PDF, 638 KB

english, 2010

11

Dithiane and trithiane-based photolabile molecular linkers equipped with amino-functionality: synthesis and quantum yields of fragmentation

Alexei N. Kurchan, Oleg D. Mitkin, Andrei G. Kutateladze

Journal:

Journal of Photochemistry and Photobiology A: Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 286 KB

english, 2005

12

Synthesis and SAR of 3-arylsulfonyl-pyrazolo[1,5-a]pyrimidines as potent serotonin 5-HT6 receptor antagonists

Alexandre V. Ivachtchenko, Elena S. Golovina, Madina G. Kadieva, Volodymyr M. Kysil, Oleg D. Mitkin, Sergey E. Tkachenko, Ilya Okun

Journal:

Bioorganic & Medicinal Chemistry

Année:

2011

Langue:

english

Fichier:

PDF, 834 KB

english, 2011

13

8-Sulfonyl-substituted tetrahydro-1H-pyrido[4,3-b]indoles as 5-HT6 receptor antagonists

Alexandre V. Ivachtchenko, Oleg D. Mitkin, Sergey E. Tkachenko, Ilya M. Okun, Volodymyr M. Kysil

Journal:

European Journal of Medicinal Chemistry

Année:

2010

Langue:

english

Fichier:

PDF, 499 KB

english, 2010

14

2-Substituted 5,6-dimethyl-3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidines: New series of highly potent and specific serotonin 5-HT6 receptor antagonists

Alexandre V. Ivachtchenko, Elena S. Golovina, Madina G. Kadieva, Angela G. Koryakova, Oleg D. Mitkin, Sergey E. Tkachenko, Volodymyr M. Kysil, Ilya Okun

Journal:

European Journal of Medicinal Chemistry

Année:

2011

Langue:

english

Fichier:

PDF, 1.04 MB

english, 2011

15

Indoles from 3-nitropyridinium salts: an extension of the transformation method on 5-substituted indoles

Oleg D Mitkin, Roman V Kombarov, Marina A Yurovskaya

Journal:

Année:

2001

Langue:

english

Fichier:

PDF, 103 KB

english, 2001

16

Solution Phase Parallel Synthesis of Substituted 3-Phenylsulfonyl-[1,2,3]triazolo[1,5-a]quinazolines: Selective Serotonin 5-HT6 Receptor Antagonists

Ivachtchenko, Alexandre V., Golovina, Elena S., Kadieva, Madina G., Koryakova, Angela G., Kovalenko, Sergiy M., Mitkin, Oleg D., Okun, Ilya M., Ravnyeyko, Irina M., Tkachenko, Sergey E., Zaremba, Oleg

Journal:

Journal of Combinatorial Chemistry

Année:

2010

Langue:

english

Fichier:

PDF, 854 KB

english, 2010

17

(3-Phenylsulfonylcycloalkano[e and d]pyrazolo[1,5-a]pyrimidin-2-yl)amines: Potent and Selective Antagonists of the Serotonin 5-HT6 Receptor

Ivachtchenko, Alexandre V., Dmitriev, Dmitri E., Golovina, Elena S., Kadieva, Madina G., Koryakova, Angela G., Kysil, Volodymyr M., Mitkin, Oleg D., Okun, Ilya M., Tkachenko, Sergey E., Vorobiev, Anto

Journal:

Journal of Medicinal Chemistry

Année:

2010

Langue:

english

Fichier:

PDF, 1.01 MB

english, 2010

18

Antagonists of 5-HT6 receptors. Substituted 3-(phenylsulfonyl)pyrazolo[1,5-a]pyrido[3,4-e]pyrimidines and 3-(phenylsulfonyl)pyrazolo[1,5-a]pyrido[4,3-d]pyrimidines—Synthesis and ‘structure–activity’ relationship

Alexandre V. Ivachtchenko, Elena S. Golovina, Madina G. Kadieva, Volodymyr M. Kysil, Oleg D. Mitkin, Anton A. Vorobiev, Ilya Okun

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2012

Langue:

english

Fichier:

PDF, 985 KB

english, 2012

19

Synthesis of substituted diphenyl sulfones and their structure–activity relationship with the antagonism of 5-НТ6 receptors

Ivachtchenko, Alexandre, Golovina, Elena, Kadieva, Madina, Mitkin, Oleg, Tkachenko, Sergei, Okun, Ilya

Journal:

Bioorganic & Medicinal Chemistry

Année:

2013

Langue:

english

Fichier:

PDF, 1.94 MB

english, 2013

20

Synthesis and Structure–Activity Relationship (SAR) of (5,7-Disubstituted 3-phenylsulfonyl-pyrazolo[1,5- a ]pyrimidin-2-yl)-methylamines as Potent Serotonin 5-HT 6 Receptor (5-HT 6 R) Antagonists

Ivachtchenko, Alexandre V., Golovina, Elena S., Kadieva, Madina G., Kysil, Volodymyr M., Mitkin, Oleg D., Tkachenko, Sergey E., Okun, Ilya M.

Journal:

Journal of Medicinal Chemistry

Année:

2011

Langue:

english

Fichier:

PDF, 1.70 MB

english, 2011

21

A novel influenza virus neuraminidase inhibitor AV5027

Ivachtchenko, Alexandre V., Ivanenkov, Yan A., Mitkin, Oleg D., Yamanushkin, Pavel M., Bichko, Vadim V., Leneva, Irina A., Borisova, Olga V.

Journal:

Antiviral Research

Année:

2013

Langue:

english

Fichier:

PDF, 1.13 MB

english, 2013

22

Dithiane- and Trithiane-Based Photolabile Scaffolds for Molecular Recognition

Mitkin, Oleg D., Kurchan, Alexei N., Wan, Yongqin, Schiwal, Brian F., Kutateladze, Andrei G.

Journal:

Organic Letters

Année:

2001

Langue:

english

Fichier:

PDF, 88 KB

english, 2001

23

Discovery of Novel Highly Potent Hepatitis C Virus NS5A Inhibitor (AV4025)

Ivachtchenko, Alexandre V., Mitkin, Oleg D., Yamanushkin, Pavel M., Kuznetsova, Irina V., Bulanova, Elena A., Shevkun, Natalia A., Koryakova, Angela G., Karapetian, Ruben N., Bichko, Vadim V., Trifele

Journal:

Journal of Medicinal Chemistry

Année:

2014

Langue:

english

Fichier:

PDF, 1.30 MB

english, 2014

24

Conical Intersection Control of Heterocyclic Photochemical Bond Scission 1,2

Zimmerman, Howard E., Mitkin, Oleg D.

Journal:

Journal of the American Chemical Society

Année:

2006

Langue:

english

Fichier:

PDF, 173 KB

english, 2006

25

Photoactive Barbiturate Receptors: An Ultimate Lock-and-Key System in Which the Key Unlocks the Lock

Lakkakula, Suman, Mitkin, Oleg D., Valiulin, Roman A., Kutateladze, Andrei G.

Journal:

Organic Letters

Année:

2007

Langue:

english

Fichier:

PDF, 89 KB

english, 2007

26

The Aza-Type-B Photochemical Rearrangement: The Role of a Second Carbonyl in Heterocyclic Photochemistry. Mechanistic and Exploratory Organic Photochemistry 1,2

Zimmerman, Howard E., Mitkin, Oleg D.

Journal:

Journal of Organic Chemistry

Année:

2007

Langue:

english

Fichier:

PDF, 115 KB

english, 2007

27

Molecular Assembly and Disassembly: Novel Photolabile Molecular Hosts

Wan, Yongqin, Mitkin, Oleg, Barnhurst, Loren, Kurchan, Alexei, Kutateladze, Andrei

Journal:

Organic Letters

Année:

2000

Langue:

english

Fichier:

PDF, 114 KB

english, 2000

28

Design, synthesis and biological evaluation of novel 5-oxo-2-thioxoimidazolidine derivatives as potent androgen receptor antagonists

Ivachtchenko, Alexandre V., Ivanenkov, Yan A., Mitkin, Oleg D., Vorobiev, Anton A., Kuznetsova, Irina V., Shevkun, Natalia A., Koryakova, Angela G., Karapetian, Ruben N., Trifelenkov, Andrey S., Kravc

Journal:

European Journal of Medicinal Chemistry

Année:

2015

Langue:

english

Fichier:

PDF, 1.35 MB

english, 2015

29

Preclinical Development of ONC1-13B, Novel Antiandrogen for Prostate Cancer Treatment

Ivachtchenko, Alexandre V., Mitkin, Oleg D., Kudan, Elizaveta V., Rjahovsky, Alexey A., Vorobiev, Anton A., Trifelenkov, Andrey S., Shevkun, Natalia A., Proskurina, Oxana V., Kravchenko, Dmitry V., Ka

Journal:

Journal of Cancer

Année:

2014

Langue:

english

Fichier:

PDF, 714 KB

english, 2014

30

Synthesis of Dithiane-Based Photolabile Molecular Systems

Mitkin, Oleg, Wan, Yongqin, Kurchan, Alexei, Kutateladze, Andrei

Journal:

Année:

2004

Langue:

english

Fichier:

PDF, 332 KB

english, 2004

31

AVN-492, A Novel Highly Selective 5-HT6R Antagonist: Preclinical Evaluation

Ivachtchenko, Alexandre V., Okun, Ilya, Aladinskiy, Vladimir, Ivanenkov, Yan, Koryakova, Angela, Karapetyan, Ruben, Mitkin, Oleg, Salimov, Ramiz, Ivashchenko, Andrey, Bezprozvanny, Ilya

Journal:

Journal of Alzheimer's Disease

Année:

2017

Langue:

english

Fichier:

PDF, 764 KB

english, 2017

32

Synthesis, X-ray crystal structure, Hirshfeld surface analysis, and molecular docking study of novel inhibitor of hepatitis B: methyl 4-fluoro-3-(morpholinosulfonyl)benzo[b]thiophene-2-carboxylate

Ivachtchenko, Alexandre V., Mitkin, Oleg D., Kravchenko, Dmitry V., Kovalenko, Sergiy M., Shishkina, Svitlana V., Bunyatyan, Natalya D., Konovalova, Irina S., Dmitrieva, Irina G., Ivanov, Vladimir V.,

Journal:

Année:

2019

Langue:

english

Fichier:

PDF, 3.12 MB

english, 2019

33

Minor C allele of the SNP rs7873784 associated with rheumatoid arthritis and type-2 diabetes mellitus binds PU.1 and enhances TLR4 expression

Korneev, Kirill V., Sviriaeva, Ekaterina N., Mitkin, Nikita A., Gorbacheva, Alisa M., Uvarova, Aksinya N., Ustiugova, Alina S., Polanovsky, Oleg L., Kulakovskiy, Ivan V., Afanasyeva, Marina A., Schwar

Journal:

Biochimica et Biophysica Acta (BBA) - Molecular Basis of Disease

Année:

2019

Langue:

english

Fichier:

PDF, 1.46 MB

english, 2019

34

Synthesis, Single Crystal X-Ray Analysis, Prediction and Study of Pharmacological Activity of 4-(1H-Benzo[d]imidazol-2-yl)-1-Phenyl-1H-1,2,3-triazol-5-Amine and Its Solvates

Ivachtchenko, Alexandre V., Mitkin, Oleg D., Kravchenko, Dmitry V., Kovalenko, Sergiy M., Shishkina, Svitlana V., Bunyatyan, Natalya D., Konovalova, Irina S., Ivanov, Vladimir V., Konovalova, Olena D.

Journal:

Année:

2019

Langue:

english

Fichier:

PDF, 4.17 MB

english, 2019

35

Minor C allele of the SNP rs7873784 associated with rheumatoid arthritis and type-2 diabetes mellitus binds PU.1 and enhances TLR4 expression

Korneev, Kirill V., Sviriaeva, Ekaterina N., Mitkin, Nikita A., Gorbacheva, Alisa M., Uvarova, Aksinya N., Ustiugova, Alina S., Polanovsky, Oleg L., Kulakovskiy, Ivan V., Afanasyeva, Marina A., Schwar

Journal:

Biochimica et Biophysica Acta (BBA) - Molecular Basis of Disease

Année:

2019

Fichier:

PDF, 1.46 MB

2019

36

Synthesis, Single Crystal X-Ray Analysis, Prediction and Study of Pharmacological Activity of 4-(1H-Benzo[d]imidazol-2-yl)-1-Phenyl-1H-1,2,3-triazol-5-Amine and Its Solvates

Ivachtchenko, Alexandre V., Mitkin, Oleg D., Kravchenko, Dmitry V., Kovalenko, Sergiy M., Shishkina, Svitlana V., Bunyatyan, Natalya D., Konovalova, Irina S., Ivanov, Vladimir V., Konovalova, Olena D.

Journal:

Année:

2019

Fichier:

PDF, 4.17 MB

2019

37

Synthesis, biological evaluation and in silico modeling of novel integrase strand transfer inhibitors (INSTIs)

Ivashchenko, Andrey A., Ivanenkov, Yan A., Koryakova, Angela G., Karapetian, Ruben N., Mitkin, Oleg D., Aladinskiy, Vladimir A., Kravchenko, Dmitry V., Savchuk, Nikolai P., Ivashchenko, Alexander V.

Journal:

European Journal of Medicinal Chemistry

Année:

2020

Fichier:

PDF, 1.45 MB

2020

38

Non-rigid Diarylmethyl Analogs of Baloxavir as CAP-Dependent Endonuclease Inhibitors of Influenza Viruses

Ivashchenko, Andrei A., Mitkin, Oleg D., Jones, Jeremy, Nikitin, Alexander V., Koryakova, Angela G., Ryakhovskiy, Alexey A., Karapetian, Ruben N., Kravchenko, Dmitry V., Aladinskiy, Vladimir, Leneva,

Journal:

Journal of Medicinal Chemistry

Année:

2020

Fichier:

PDF, 1.16 MB

2020